Get 20M+ Full-Text Papers For Less Than $1.50/day. Start a 14-Day Trial for You or Your Team.

Learn More →

Copper‐Mediated Direct and Selective C−H Thiolation of Quinazolinones

Copper‐Mediated Direct and Selective C−H Thiolation of Quinazolinones Direct thiolation of quinazolinones by selective cleavage of a relatively inert C−H bond, mediated by earth‐abundant copper and guided by a pyridine or pyrimidine moiety, has been achieved under operationally simple conditions. The devised protocol does not require any toxic or reactive reagents and provides direct access to a broad spectrum of pharmaceutically relevant thioquinazolinones. http://www.deepdyve.com/assets/images/DeepDyve-Logo-lg.png Asian Journal of Organic Chemistry Wiley

Copper‐Mediated Direct and Selective C−H Thiolation of Quinazolinones

Loading next page...
 
/lp/wiley/copper-mediated-direct-and-selective-c-h-thiolation-of-quinazolinones-BjxiqevvuC

References (74)

Publisher
Wiley
Copyright
© 2019 Wiley‐VCH Verlag GmbH & Co. KGaA, Weinheim
ISSN
2193-5807
eISSN
2193-5815
DOI
10.1002/ajoc.201900199
Publisher site
See Article on Publisher Site

Abstract

Direct thiolation of quinazolinones by selective cleavage of a relatively inert C−H bond, mediated by earth‐abundant copper and guided by a pyridine or pyrimidine moiety, has been achieved under operationally simple conditions. The devised protocol does not require any toxic or reactive reagents and provides direct access to a broad spectrum of pharmaceutically relevant thioquinazolinones.

Journal

Asian Journal of Organic ChemistryWiley

Published: Jun 1, 2019

Keywords: ; ; ; ;

There are no references for this article.