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Direct thiolation of quinazolinones by selective cleavage of a relatively inert C−H bond, mediated by earth‐abundant copper and guided by a pyridine or pyrimidine moiety, has been achieved under operationally simple conditions. The devised protocol does not require any toxic or reactive reagents and provides direct access to a broad spectrum of pharmaceutically relevant thioquinazolinones.
Asian Journal of Organic Chemistry – Wiley
Published: Jun 1, 2019
Keywords: ; ; ; ;
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